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Charles Henley Selected Research

N- (2- chlorophenylpropyl)- 1- (3- methoxyphenyl)ethylamine

11/2009Discovery and optimization of substituted 1-(1-phenyl-1H-pyrazol-3-yl)methanamines as potent and efficacious type II calcimimetics.
8/2009R-568 reduces ectopic calcification in a rat model of chronic kidney disease-mineral bone disorder (CKD-MBD).
7/2009Calcimimetic inhibits late-stage cyst growth in ADPKD.

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Charles Henley Research Topics

Disease

6Secondary Hyperparathyroidism
12/2013 - 07/2005
3Chronic Renal Insufficiency
06/2011 - 07/2005
2Hypercalcemia (Milk Alkali Syndrome)
07/2013 - 03/2011
2Chronic Kidney Disease-Mineral and Bone Disorder (Renal Rickets)
07/2012 - 08/2009
2Vascular Calcification
08/2009 - 07/2005
1Bone Resorption
07/2013
1Neoplasms (Cancer)
07/2013
1Hypophosphatemia
07/2013
1Hypocalcemia
06/2011
1Thyroid Neoplasms (Thyroid Cancer)
06/2011
1Hyperplasia
08/2009
1Bone Diseases (Bone Disease)
08/2009
1Uremia
08/2009
1Hyperparathyroidism
08/2009
1Fibrosis (Cirrhosis)
07/2009
1Polycystic Kidney Diseases (Polycystic Kidney Disease)
07/2009
1Disease Progression
07/2009
1Cysts
07/2009
1Alzheimer Disease (Alzheimer's Disease)
10/2007
1Pain (Aches)
10/2007
1Hyperthermia
10/2007
1Ischemic Stroke
10/2007
1Amyotrophic Lateral Sclerosis (Lou Gehrig's Disease)
10/2007
1Neurodegenerative Diseases (Neurodegenerative Disease)
10/2007

Drug/Important Bio-Agent (IBA)

5CalciumIBA
07/2013 - 07/2005
4Phosphorus (Red Phosphorus)IBA
07/2013 - 07/2005
4Parathyroid Hormone (Parathormone)IBA
08/2009 - 07/2005
3Cinacalcet (Sensipar)FDA Link
07/2013 - 07/2005
3N- (2- chlorophenylpropyl)- 1- (3- methoxyphenyl)ethylamineIBA
11/2009 - 07/2009
2Calcitonin (Calcitonin, Eel)FDA LinkGeneric
07/2013 - 06/2011
2Calcium-Sensing ReceptorsIBA
07/2013 - 07/2009
2MineralsIBA
07/2012 - 08/2009
2N- ((6- (methyloxy)- 4'- (trifluoromethyl)- 3- biphenylyl)methyl)- 1- phenylethanamineIBA
03/2011 - 08/2009
2Calcitriol (Calcijex)FDA LinkGeneric
08/2009 - 07/2005
1Urea (Carbamide)FDA LinkGeneric
12/2013
1Ribonucleases (Ribonuclease)IBA
07/2013
1Messenger RNA (mRNA)IBA
07/2013
1Parathyroid Hormone-Related ProteinIBA
07/2013
1Type 1 Parathyroid Hormone Receptor (Parathyroid Hormone Receptor)IBA
07/2013
1Hormones (Hormone)IBA
07/2012
1Phosphates (Orthophosphate)IBA
07/2012
1Calcimimetic AgentsIBA
11/2009
1Vitamin DFDA LinkGeneric
08/2009
1AdenineFDA LinkGeneric
08/2009
1SterolsIBA
08/2009
1polycystic kidney disease 1 proteinIBA
07/2009
1Capsaicin (Zostrix)FDA Link
10/2007
1TRPV Cation ChannelsIBA
10/2007
1Cyclin-Dependent Kinase 5IBA
10/2007
1N- (4- (6- (4- trifluoromethylphenyl)pyrimidin- 4- yloxy)benzothiazol- 2- yl)acetamideIBA
10/2007
1Protein Serine-Threonine Kinases (Protein-Serine-Threonine Kinase)IBA
10/2007
1AntipyreticsIBA
10/2007
1Acetaminophen (Paracetamol)FDA LinkGeneric
10/2007
1CationsIBA
10/2007

Therapy/Procedure

1Therapeutics
10/2007